SCHEMBL5573239

SCHEMBL5573239

CCOC(=O)[C@H](O)Cc1cc(C)c2[nH]ncc2c1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
HIF1A Q16665 1/20 0.41
CALCA P06881 8/20 0.41
CALCRL Q16602 6/20 0.38
ACACB O00763 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22796661 0.90 CALCA (0.40) CALCACALCRL
SCHEMBL28708104 0.90 CALCA (0.40) CALCACALCRL
SCHEMBL29549510 0.86 ACACB (0.43) CALCACALCRLACACB
SCHEMBL29996805 0.86 ACACB (0.43) CALCACALCRLACACB
SCHEMBL28704453 0.86 ACACB (0.43) CALCACALCRLACACB
SCHEMBL22796477 0.86 ACACB (0.43) CALCACALCRLACACB
SCHEMBL3353840 0.85 CALCA (0.41) CALCACALCRL
SCHEMBL3353834 0.85 CALCA (0.41) CALCACALCRL
SCHEMBL107000 0.79 CALCA (0.39) CALCACALCRL
SCHEMBL22796447 0.79 CALCA (0.39) CALCACALCRL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740577-A2 SELECTED CGRP ANTAGONISTS, METHODS FOR THE PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-01-10 EP disclosed
WO-2005103037-A2 SELECTED CGRP ANTAGONISTS, METHODS FOR THE PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-03 WO disclosed