SCHEMBL5574155

SCHEMBL5574155

CC(C)N(/C=N/c1ncc(C#Cc2ccc(Cl)cc2)c(Nc2ccc(O)cc2)n1)C(C)C

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AURKA O14965 5/20 0.36
GAA P10253 2/20 0.32
TP53 P04637 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
VCP P55072 1/20 0.32
APP P05067 1/20 0.32
GRM5 P41594 1/20 0.31
FGFR1 P11362 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3251691 1.00 AURKA (0.36) AURKAGAATP53POLBMAPT
SCHEMBL3248475 0.81 KDM4E (0.33) GRM5
SCHEMBL3254180 0.79 MERTK (0.34)
SCHEMBL3254181 0.79 MERTK (0.34)
SCHEMBL3254176 0.79 MERTK (0.34)
SCHEMBL3251095 0.75 AURKA (0.45) AURKAGAATP53POLBMAPT
SCHEMBL3254024 0.72 PLAU (0.34) GRM5
SCHEMBL3248012 0.72 ADK (0.42) GAAMAPT
SCHEMBL3264002 0.71 ADK (0.39) MAPT
SCHEMBL3251683 0.71 ACACB (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7205297-B2 Substituted 5-alkynyl pyrimidines having neurotrophic activity KRENITSKY PHARMACEUTICALS, INC. (US) 2007-04-17 US disclosed