SCHEMBL5575175

SCHEMBL5575175

O=C(O)C(Cc1ccc(Nc2nccc3ccncc23)cc1)NC1=CC(=O)C12CCCCC2

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 20/20 0.55
ITGA4 P13612 20/20 0.55
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2978998 1.00 ITGB1 (0.55) ITGB1ITGA4CYP3A4CYP2C9
SCHEMBL3832796 0.90 ITGB1 (0.47) ITGB1ITGA4CYP3A4CYP2C9
SCHEMBL2980605 0.89 ITGA4 (0.54) ITGB1ITGA4CYP3A4CYP2C9
Zaurategrast SCHEMBL5571298 0.86 ITGB1 (0.56) ITGB1ITGA4CYP3A4CYP2C9
Zaurategrast SCHEMBL2976322 0.86 ITGB1 (0.56) ITGB1ITGA4CYP3A4CYP2C9
SCHEMBL2974021 0.84 ITGB1 (0.54) ITGB1ITGA4CYP3A4CYP2C9
SCHEMBL7265369 0.84 ITGB1 (0.54) ITGB1ITGA4CYP3A4CYP2C9
SCHEMBL2990251 0.84 ITGB1 (0.56) ITGB1ITGA4CYP3A4CYP2C9
SCHEMBL3832798 0.82 ITGB1 (0.38) ITGB1ITGA4
SCHEMBL6131672 0.82 ITGB1 (0.38) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1780201-A2 PHENYLALANINE ENAMIDE DERIVATIVES POSSESSING A CYCLOBUTENE GROUP, FOR USE AS INTEGRIN INHIBITORS Celltech R&D Limited (GB) 2007-05-02 EP disclosed
EP-1370531-B1 PHENYLALANINE ENAMIDE DERIVATIVES POSSESSING A CYCLOBUTENE GROUP, FOR USE AS INTEGRIN INHIBITORS CELLTECH R&D LTD (GB) 2007-02-28 EP disclosed