SCHEMBL5576013

SCHEMBL5576013

Cc1cnc(CNCCCCNCc2nccc3ccccc23)c(C)c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ADORA2A P29274 2/20 0.37
CHRM2 P08172 2/20 0.37
MAPK1 P28482 1/20 0.37
SLC40A1 Q9NP59 1/20 0.36
F2 P00734 1/20 0.36
F10 P00742 1/20 0.36
SCN8A Q9UQD0 2/20 0.36
CYP1A2 P05177 1/20 0.34
SLC2A1 P11166 1/20 0.34
CXCR4 P61073 1/20 0.34
ROCK1 Q13464 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5576002 0.88 CXCR4 (0.37) CYP2A6MEN1KMT2AADORA2ACHRM2
SCHEMBL2084845 0.78 TMEM97 (0.38) CYP2A6CHRM2MAPK1CXCR4
SCHEMBL2084170 0.77 CXCR4 (0.41) CYP2A6CHRM2CXCR4
SCHEMBL11935014 0.77 CHRM2 (0.45) ADORA2ACHRM2CYP1A2CXCR4ADORA1
SCHEMBL2080968 0.75 CXCR4 (0.39) CYP2A6MEN1KMT2AADORA2ACHRM2
SCHEMBL2311388 0.75 PLAU (0.48) CYP2A6MEN1KMT2AADORA2AMAPK1
SCHEMBL23398172 0.74 CXCR4 (0.42) MEN1KMT2AADORA2ACHRM2SLC40A1
SCHEMBL2084248 0.74 TP53 (0.38) KMT2AADORA2ACHRM2MAPK1SLC40A1
SCHEMBL30482129 0.72 CYP2A6 (0.47) CYP2A6MEN1KMT2AADORA2AMAPK1
SCHEMBL7334545 0.72 CYP2A6 (0.47) CYP2A6MEN1KMT2AADORA2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7291631-B2 CXCR4 chemokine receptor binding compounds GENZYME CORPORATION (US) 2007-11-06 US disclosed
US-20040209921-A1 CXCR4 chemokine receptor binding comounds ANORMED CORPORATION (CA) 2004-10-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040209921-A1 CXCR4 chemokine receptor binding comounds CXCR4, CXCR1, CXCR3 CYP2A6 3010/4885MEN1 4472/4885KMT2A 4082/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.