SCHEMBL5576797

SCHEMBL5576797

CCCCOC(=O)N1CC2c3cc(CCC)cc(Cl)c3C(=O)N(C)C2C1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 8/20 0.45
HTR2C P28335 8/20 0.45
HTR2B P41595 8/20 0.45
DPP4 P27487 1/20 0.36
LMNA P02545 2/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
OPRK1 P41145 1/20 0.32
ESR1 P03372 1/20 0.32
ENPP2 Q13822 2/20 0.31
HRH2 P25021 1/20 0.31
HRH1 P35367 1/20 0.31
ALDH1A1 P00352 2/20 0.30
TSHR P16473 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
THRB P10828 1/20 0.30
KMT2A Q03164 1/20 0.30
SMYD3 Q9H7B4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4473909 0.86 HTR2A (0.46) HTR2AHTR2CHTR2BDPP4
SCHEMBL4483372 0.85 HTR2A (0.51) HTR2AHTR2CHTR2BDPP4POLB
SCHEMBL13763136 0.78 HTR2A (0.55) HTR2AHTR2CHTR2B
SCHEMBL13756865 0.72 HTR2C (0.82) HTR2AHTR2CHTR2B
SCHEMBL13756868 0.72 HTR2C (0.82) HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL4467012 0.71 HTR2A (0.83) HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL4472459 0.71 HTR2A (0.83) HTR2AHTR2CHTR2B
SCHEMBL13756911 0.70 HTR2A (0.68) HTR2AHTR2CHTR2BLMNAALDH1A1
Hydrochloric Acid SCHEMBL4467773 0.69 HTR2A (0.69) HTR2AHTR2CHTR2BLMNAALDH1A1
SCHEMBL13763057 0.69 HTR2A (0.67) HTR2AHTR2CHTR2BLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778225-A2 PYRROLO(OXO)ISOQUINOLINES AS 5HT LIGANDS Bristol-Myers Squibb Company (US) 2007-05-02 EP disclosed
WO-2006019886-A2 PYRROLO(OXO)ISOQUINOLINES AS 5HT LIGANDS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-02-23 WO disclosed