SCHEMBL5576980

SCHEMBL5576980

Cc1ccc(CC(N)CCCNC(C)c2ccccn2)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 5/20 0.46
P2RX3 P56373 1/20 0.41
SCN8A Q9UQD0 2/20 0.37
TLR7 Q9NYK1 2/20 0.34
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
MAPK1 P28482 1/20 0.31
CHRM2 P08172 2/20 0.30
CHRM4 P08173 2/20 0.30
CHRM5 P08912 2/20 0.30
CHRM1 P11229 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5574432 0.83 CXCR4 (0.48) CXCR4P2RX3SCN8ATLR7MAPK1
SCHEMBL5576630 0.76 SCN8A (0.35) CXCR4SCN8ATLR7EGFR
SCHEMBL2083756 0.76 CXCR4 (0.53) CXCR4P2RX3TLR7HDAC1HDAC2
SCHEMBL20278941 0.71 NOS3 (0.37) CXCR4P2RX3TLR7HDAC6
SCHEMBL12812606 0.68 KCNA5 (0.49) SCN8ACHRM2CHRM1EGFR
SCHEMBL22894779 0.67 CYP1A2 (0.58)
SCHEMBL30894457 0.67 CHRM2 (0.62) SCN8AGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL20031861 0.66 NOS3 (0.41) CXCR4TLR7HDAC6
SCHEMBL1968196 0.66 NOS3 (0.41) CXCR4TLR7HDAC6CHRM2CHRM4
SCHEMBL15131054 0.66 SLC6A2 (0.65) CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7291631-B2 CXCR4 chemokine receptor binding compounds GENZYME CORPORATION (US) 2007-11-06 US claimed