Guanine

Guanine

SCHEMBL5579240

Nc1cc[nH]c(=O)n1.Nc1nc2nc[nH]c2c(=O)[nH]1.O=c1cc[nH]c(=O)[nH]1

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PNP P00491 2/20 0.60
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CRBN Q96SW2 1/20 0.40
GRIA1 P42261 1/20 0.39
GRIA2 P42262 1/20 0.39
GRIA3 P42263 1/20 0.39
GRIA4 P48058 1/20 0.39
GDA Q9Y2T3 1/20 0.38
DYRK1A Q13627 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Guanine SCHEMBL2636587 0.92 PNP (0.51) PNPKDM4EMEN1ALDH1A1MAPT
Guanine SCHEMBL2499473 0.92 PNP (0.72) PNPKDM4EMEN1ALDH1A1MAPT
Guanine SCHEMBL79001 0.92 PNP (0.72) PNPKDM4EMEN1ALDH1A1MAPT
Guanine SCHEMBL2528337 0.92 PNP (0.72) PNPKDM4EMEN1ALDH1A1MAPT
Guanine SCHEMBL2529420 0.92 PNP (0.72) PNPKDM4EMEN1ALDH1A1MAPT
Guanine SCHEMBL23576542 0.86 PNP (0.63) PNPKDM4EMEN1ALDH1A1MAPT
Guanine SCHEMBL19991865 0.85 PNP (0.62) PNPKDM4EMEN1ALDH1A1MAPT
Guanine SCHEMBL15718981 0.85 PNP (0.43) PNPKDM4EMEN1ALDH1A1MAPT
Guanine SCHEMBL20518478 0.84 PNP (0.55) PNPKDM4EMEN1ALDH1A1MAPT
Guanine SCHEMBL23880590 0.84 PNP (0.55) PNPKDM4EMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2500437-B1 Methods for identifying compounds that modulate untranslated region-dependent gene expression and methods of using same PTC THERAPEUTICS INC (US) 2016-11-30 EP disclosed
US-9493845-B2 Methods for identifying compounds that modulate untranslated region-dependent gene expression and methods of using same PTC THERAPEUTICS, INC. (US) 2016-11-15 US disclosed
US-8618077-B2 Compositions and methods for treating fragile X premutation RVGG repeats-mediated toxicity EMORY UNIVERSITY (US) 2013-12-31 US disclosed
US-20130347133-A1 Methods For Identifying Compounds That Modulate Untranslated Region-Dependent Gene Expression And Methods Of Using Same PTC THERAPEUTICS, INC. (US) 2013-12-26 US disclosed
US-8460864-B2 Methods for identifying compounds that modulate untranslated region-dependent gene expression and methods of using same PTC THERAPEUTICS, INC. (US) 2013-06-11 US disclosed
US-20120277178-A1 COMPOSITIONS AND METHODS FOR TREATING FRAGILE X PREMUTATION RVGG REPEATS-MEDIATED TOXICITY EMORY UNIVERSITY (US) 2012-11-01 US disclosed
EP-2500437-A2 Methods for identifying compounds that modulate untranslated region-dependent gene expression and methods of using same PTC Therapeutics, Inc. (US) 2012-09-19 EP disclosed
US-20070111203-A1 Methods for identifying compounds that modulate untranslated region-dependent gene expression and methods of using same PTC THERAPEUTICS 2007-05-17 US disclosed