SCHEMBL5579585

SCHEMBL5579585

CCc1cccc(CNCC(OC(=O)CCC(=O)Nc2nnc(-c3ccccc3)s2)C(N)Cc2cc(F)cc(F)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
BACE1 P56817 9/20 0.38
CTSB P07858 7/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CTSD P07339 2/20 0.36
PRKACA P17612 1/20 0.36
ROCK1 Q13464 1/20 0.36
NOX1 Q9Y5S8 1/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5579577 1.00 KDM4E (0.41) KDM4EALDH1A1HPGDHSD17B10BACE1
SCHEMBL5579493 0.91 CYP1A2 (0.47) KDM4EALDH1A1HSD17B10NPC1RAB9A
SCHEMBL5579494 0.91 CYP1A2 (0.47) KDM4EALDH1A1HSD17B10NPC1RAB9A
SCHEMBL5126861 0.91 BACE1 (0.38) ALDH1A1BACE1CTSBNPC1SMN1; SMN2
SCHEMBL5579505 0.86 KMT2A (0.38) ALDH1A1HSD17B10BACE1CTSBSMN1; SMN2
SCHEMBL5579513 0.86 KMT2A (0.38) ALDH1A1HSD17B10BACE1CTSBSMN1; SMN2
SCHEMBL5124419 0.82 KMT2A (0.42) BACE1CTSBKMT2ACTSDHDAC1
SCHEMBL5124411 0.82 KMT2A (0.42) BACE1CTSBKMT2ACTSDHDAC1
SCHEMBL3346887 0.82 BACE1 (0.52) BACE1CTSBCTSD
SCHEMBL13308143 0.82 BACE1 (0.52) BACE1CTSBCTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7294642-B2 1,3-Diamino-2-hydroxypropane pro-drug derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-11-13 US claimed