SCHEMBL5579589

SCHEMBL5579589

CCC[C@](N)(SCC(=O)Nc1ccc(-c2cnco2)c(-c2cc(F)cc(F)c2)c1)C(=O)OCNCc1cccc(CC)c1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 10/20 0.38
AAK1 Q2M2I8 10/20 0.38
IMPDH1 P20839 5/20 0.36
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5130670 0.89 BACE1 (0.39) IMPDH2AAK1
SCHEMBL5579814 0.69 BACE1 (0.33)
SCHEMBL3350514 0.65 BACE1 (0.47)
SCHEMBL13308180 0.65 BACE1 (0.47)
SCHEMBL5377505 0.65 BACE1 (0.47)
SCHEMBL5377510 0.65 BACE1 (0.47)
SCHEMBL5579586 0.65 AAK1 (0.37) IMPDH2AAK1IMPDH1
SCHEMBL5579592 0.65 AAK1 (0.37) IMPDH2AAK1IMPDH1
SCHEMBL5579599 0.65 AAK1 (0.37) IMPDH2AAK1IMPDH1
SCHEMBL5579545 0.65 BACE1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7294642-B2 1,3-Diamino-2-hydroxypropane pro-drug derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-11-13 US claimed