SCHEMBL5579899

SCHEMBL5579899

CCc1nc2ccccc2n1OC(C)=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
KMT2A Q03164 1/20 0.46
TSHR P16473 2/20 0.44
MAPK1 P28482 2/20 0.44
RECQL P46063 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
APEX1 P27695 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TP53 P04637 1/20 0.44
CASP1 P29466 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3968907 0.79 TSHR (0.52) CYP1A2CYP3A4CYP2D6KDM4EALDH1A1
SCHEMBL12473755 0.78 SMN1; SMN2 (0.51) CYP1A2CYP3A4CYP2D6KDM4EALDH1A1
SCHEMBL27697871 0.74 PTGDR2 (0.61) ALDH1A1MEN1MAPTKMT2ATSHR
SCHEMBL6946448 0.73 TSHR (0.49) CYP1A2CYP3A4CYP2D6KDM4EALDH1A1
SCHEMBL29145189 0.73 L3MBTL1 (0.61) CYP1A2CYP3A4CYP2D6KDM4EALDH1A1
SCHEMBL18955291 0.71 APEX1 (0.73) KDM4EALDH1A1MEN1HPGDKMT2A
SCHEMBL17627891 0.71 KDM4E (0.52) CYP1A2CYP3A4KDM4EALDH1A1MEN1
SCHEMBL31596375 0.71 APEX1 (0.73) KDM4EALDH1A1MEN1HPGDKMT2A
SCHEMBL13776647 0.70 TSHR (0.51) CYP1A2CYP3A4CYP2D6KDM4EALDH1A1
SCHEMBL14300652 0.70 CYP1A2 (0.46) CYP1A2CYP3A4CYP2D6KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7294642-B2 1,3-Diamino-2-hydroxypropane pro-drug derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-11-13 US claimed