SCHEMBL5583496

SCHEMBL5583496

CC(=O)Nc1ccccc1OCC(C)(O)CN(Cc1ccc(F)c(F)c1)C1CCNCC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.46
SLC6A4 P31645 9/20 0.40
SLC6A2 P23975 9/20 0.40
HTR6 P50406 1/20 0.39
CCR1 P32246 1/20 0.38
BRD4 O60885 2/20 0.38
SLC6A3 Q01959 6/20 0.37
SSTR4 P31391 1/20 0.36
MAPK14 Q16539 1/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MRGPRX1 Q96LB2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5583430 0.93 ABCB11 (0.48) ABCB11SLC6A4SLC6A2CCR1BRD4
SCHEMBL7263208 0.89 ABCB11 (0.58) ABCB11SLC6A4SLC6A2CCR1BRD4
SCHEMBL5583485 0.89 ABCB11 (0.58) ABCB11SLC6A4SLC6A2CCR1BRD4
SCHEMBL5583417 0.89 ABCB11 (0.48) ABCB11SLC6A4SLC6A2HTR6CCR1
SCHEMBL5583514 0.87 ABCB11 (0.48) ABCB11SLC6A4SLC6A2CCR1BRD4
SCHEMBL5583488 0.83 ABCB11 (0.46) ABCB11SLC6A4SLC6A2CCR1SLC6A3
Benzoic Acid SCHEMBL4199385 0.79 CCR1 (0.54) ABCB11SLC6A4SLC6A2CCR1BRD4
SCHEMBL4199387 0.78 CCR1 (0.45) ABCB11SLC6A4SLC6A2CCR1BRD4
SCHEMBL7264055 0.76 ABCB11 (0.47) ABCB11SLC6A4SLC6A2CCR1SLC6A3
SCHEMBL7268791 0.74 SLC6A2 (0.52) ABCB11SLC6A4SLC6A2CCR1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4022142-B2 2007-12-12 JP claimed
JP-2004507461-A 2004-03-11 JP claimed
EP-1299357-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2003-04-09 EP claimed
WO-2001098273-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2001-12-27 WO claimed
EP-1299357-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2003-04-09 EP disclosed
WO-2001098273-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2001-12-27 WO disclosed