SCHEMBL5586148

SCHEMBL5586148

Cc1cccc(-c2noc(NC(=O)Cc3cccc(F)c3F)c2-c2ccncn2)c1

nearest known ligand 0.77

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 16/20 0.77
MAPK9 P45984 1/20 0.58
MAPK10 P53779 1/20 0.58
MAPK11 Q15759 1/20 0.58
MLYCD O95822 1/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
CXCR2 P25025 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1881717 0.94 MAPK14 (0.81) MAPK14MAPK9MAPK10MAPK11LMNA
SCHEMBL1882588 0.89 MAPK14 (0.73) MAPK14MAPK9MAPK10MAPK11MEN1
SCHEMBL1882291 0.89 MAPK14 (0.73) MAPK14MAPK9MAPK10MAPK11MEN1
SCHEMBL1872761 0.89 MAPK14 (0.84) MAPK14MAPK9MAPK10MAPK11
SCHEMBL5586103 0.88 MAPK14 (0.79) MAPK14MAPK9MAPK10MAPK11
SCHEMBL1881306 0.87 MAPK14 (0.81) MAPK14MAPK9MAPK10MAPK11
SCHEMBL1877324 0.87 MAPK14 (1.00) MAPK14MAPK9MAPK10MAPK11
SCHEMBL1877548 0.87 MAPK14 (0.81) MAPK14MAPK9MAPK10MAPK11
SCHEMBL1877611 0.87 MAPK14 (0.78) MAPK14MAPK9MAPK10MAPK11
SCHEMBL1882877 0.87 MAPK14 (0.79) MAPK14MAPK9MAPK10MAPK11MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1832584-A1 PYRIMIDINYLISOXAZOL DERIVATIVE ASKA Pharmaceutical Co., Ltd. (JP) 2007-09-12 EP disclosed