SCHEMBL5593757

SCHEMBL5593757

Cc1cc2[nH]nc(C3CC3c3ccccc3)c2cc1NC(=O)Cc1ccc(N(C)C)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 4/20 0.51
AURKB Q96GD4 3/20 0.46
CDK2 P24941 3/20 0.42
CDK1 P06493 1/20 0.41
CDK4 P11802 1/20 0.41
EPHX2 P34913 1/20 0.40
CACNA1G O43497 3/20 0.39
CACNA1H O95180 3/20 0.39
CACNA1I Q9P0X4 3/20 0.39
GSK3B P49841 1/20 0.39
GLS O94925 1/20 0.38
FLT3 P36888 1/20 0.38
KDM1A O60341 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HPGD P15428 1/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
KCNH2 Q12809 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5594175 0.87 AURKA (0.58) AURKAAURKBCDK2CDK1CDK4
SCHEMBL14539029 0.80 AURKA (0.39) AURKAAURKBGSK3BSMN1; SMN2
SCHEMBL5594098 0.77 AURKA (0.68) AURKAAURKBCDK2CDK1CDK4
SCHEMBL14538838 0.73 AURKA (0.58) AURKAAURKBCDK2CDK1CDK4
SCHEMBL4495289 0.70 GSK3B (0.73) AURKBCDK2CDK1CDK4GSK3B
SCHEMBL5867743 0.63 CDK2 (0.45) CDK2CDK1CDK4CACNA1GCACNA1H
SCHEMBL22890624 0.62 LRRK2 (0.74)
SCHEMBL22890323 0.62 LRRK2 (0.74)
SCHEMBL29643542 0.62 LRRK2 (0.74)
SCHEMBL6390395 0.61 CDK2 (0.47) CDK2CDK1CDK4CACNA1GCACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007058626-A1 INDAZOLE COMPOUNDS S*BIO PTE LTD (SG) 2007-05-24 WO claimed