SCHEMBL5598008

SCHEMBL5598008

Nc1ccc2c(c1)C(c1ccccc1)=NCCN2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 4/20 0.44
CHRM1 P11229 5/20 0.40
ALDH1A1 P00352 2/20 0.40
CNR1 P21554 1/20 0.40
NTSR1 P30989 1/20 0.40
OPRK1 P41145 1/20 0.40
PDE4D Q08499 1/20 0.40
PKM P14618 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
KDM4E B2RXH2 2/20 0.39
MEN1 O00255 2/20 0.39
NPC1 O15118 2/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
USP2 O75604 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1199602 0.82 CHRM1 (0.59) NISCHCHRM1ALDH1A1CNR1NTSR1
SCHEMBL12876624 0.82 CHRM1 (0.59) NISCHCHRM1CNR1NTSR1OPRK1
SCHEMBL29414926 0.82 CHRM1 (0.59) NISCHCHRM1ALDH1A1CNR1NTSR1
SCHEMBL11460470 0.82 CHRM1 (0.59) NISCHCHRM1ALDH1A1CNR1NTSR1
SCHEMBL1199345 0.81 NISCH (0.54) NISCHADRA2AADRA2BADRA2C
SCHEMBL1198373 0.80 KDM4E (0.50) NISCHCHRM1ALDH1A1CNR1NTSR1
SCHEMBL11678875 0.79 CHRM1 (0.62) NISCHCHRM1ALDH1A1CNR1NTSR1
SCHEMBL12707822 0.79 NISCH (0.41) NISCHALDH1A1KDM4EMEN1NPC1
SCHEMBL11852207 0.79 KDM4E (0.43) NISCHALDH1A1CNR1NTSR1OPRK1
SCHEMBL1199546 0.79 AURKA (0.50) NISCHALDH1A1KDM4EMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007072041-A1 THERAPEUTIC COMPOUNDS ASTEX THERAPEUTICS LIMITED (GB) 2007-06-28 WO disclosed