SCHEMBL5604086

SCHEMBL5604086

CC1CC(N)c2ncccc2O1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.32
LTA4H P09960 1/20 0.31
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31
CHRNB4 P30926 2/20 0.31
CHRNA3 P32297 2/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNA4 P43681 1/20 0.31
PRKCA P17252 1/20 0.30
PRKCQ Q04759 1/20 0.30
AKR1B1 P15121 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30630775 1.00 CYP2A6 (0.32) CYP2A6LTA4HBRD4CREBBPCHRNB4
SCHEMBL14136494 0.79 CHRNB4 (0.33) LTA4HBRD4CREBBPCHRNB4CHRNA3
Hydrochloric Acid SCHEMBL27094825 0.74 MEN1 (0.31) CYP2A6PRKCAPRKCQ
SCHEMBL26625675 0.72 BRD4 (0.33) BRD4CREBBPCHRNB4CHRNA3CHRNB2
SCHEMBL27094529 0.72 AKR1B1 (0.39) LTA4HAKR1B1
SCHEMBL14661123 0.72 LTA4H (0.40) LTA4HCHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL1328841 0.72 POLB (0.43) BRD4CREBBPAKR1B1
SCHEMBL18383187 0.72 POLB (0.43) BRD4CREBBPAKR1B1
SCHEMBL18383190 0.72 POLB (0.43) BRD4CREBBPAKR1B1
SCHEMBL23219887 0.70 LTA4H (0.31) LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1838312-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-10-03 EP disclosed
WO-2006076131-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-07-20 WO disclosed