SCHEMBL5606019

SCHEMBL5606019

Cc1cc2c(c(-c3cc(Cl)ccc3Cl)c1)OC(C(C)N)C2

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 2/20 0.37
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
HTT P42858 1/20 0.31
EZH2 Q15910 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
S1PR4 O95977 2/20 0.30
HTR2A P28223 2/20 0.30
HTR2C P28335 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5605407 0.90 AQP1 (0.47) AQP1LMNATP53HTTEZH2
SCHEMBL5605912 0.85 AQP1 (0.35) AQP1LMNAKDM4EALDH1A1MAPT
SCHEMBL6048001 0.82 S1PR4 (0.35) AQP1LMNAKDM4EALDH1A1MAPT
SCHEMBL4766477 0.81 AQP1 (0.39) AQP1LMNAKDM4EALDH1A1MAPT
SCHEMBL4766472 0.80 AQP1 (0.38) AQP1KDM4EALDH1A1MAPTS1PR4
SCHEMBL4220746 0.79 AQP1 (0.60) AQP1EZH2KDM4EALDH1A1MAPT
SCHEMBL5606024 0.78 AQP1 (0.37) AQP1LMNAKDM4EALDH1A1MAPT
SCHEMBL4220770 0.77 AQP1 (0.49) AQP1EZH2ALDH1A1S1PR4
SCHEMBL4220767 0.75 AQP1 (0.64) AQP1EZH2KDM4EALDH1A1MAPT
SCHEMBL4790052 0.75 AQP1 (0.44) AQP1EZH2S1PR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007509174-A 2007-04-12 JP claimed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP claimed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO claimed