SCHEMBL5607804

SCHEMBL5607804

Cc1cc(C)c(NC(=O)c2sc(NCCC(=O)c3ccccc3)nc2C)c(C)c1

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LCK P06239 15/20 0.71
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
ALDH1A1 P00352 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5608004 0.94 LCK (0.69) LCKNPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL5607823 0.88 LCK (0.58) LCKNPC1RAB9A
SCHEMBL3720281 0.85 LCK (0.61) LCKNPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL5607634 0.84 LCK (0.56) LCKNPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL773819 0.83 LCK (1.00) LCKNPC1RAB9ASMN1; SMN2
SCHEMBL7626148 0.82 LCK (0.69) LCK
SCHEMBL773079 0.82 LCK (0.64) LCKNPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL5608106 0.81 LCK (0.52) LCKNPC1RAB9AALDH1A1SMN1; SMN2
Benzene SCHEMBL773080 0.81 LCK (0.69) LCKNPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL3719150 0.79 LCK (0.54) LCKNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758564-A2 SYNERGISTIC METHODS AND COMPOSITIONS FOR TREATING CANCER Brystol-Myers Squibb Company (US) 2007-03-07 EP claimed
WO-2005094376-A2 SYNERGISTIC METHODS AND COMPOSITIONS FOR TREATING CANCER BRISTOL-MYERS SQUIBB COMPANY (US) 2005-10-13 WO claimed
EP-1758564-A2 SYNERGISTIC METHODS AND COMPOSITIONS FOR TREATING CANCER Brystol-Myers Squibb Company (US) 2007-03-07 EP disclosed
WO-2005094376-A2 SYNERGISTIC METHODS AND COMPOSITIONS FOR TREATING CANCER BRISTOL-MYERS SQUIBB COMPANY (US) 2005-10-13 WO disclosed