SCHEMBL5609308

SCHEMBL5609308

COc1ccc(N(c2ccc(N(C)C)cc2)c2cccc(C)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.49
SLC2A1 P11166 1/20 0.49
ACHE P22303 2/20 0.47
NPC1 O15118 5/20 0.45
RAB9A P51151 5/20 0.45
TDP1 Q9NUW8 2/20 0.45
RELA Q04206 2/20 0.45
MEN1 O00255 1/20 0.45
NSD2 O96028 1/20 0.45
CASP3 P42574 1/20 0.45
KMT2A Q03164 1/20 0.45
SENP8 Q96LD8 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
MAPT P10636 4/20 0.43
TP53 P04637 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
ALDH1A1 P00352 2/20 0.43
ESR2 Q92731 1/20 0.43
NOX1 Q9Y5S8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14158330 0.93 ACHE (0.53) ACHENPC1RAB9ATDP1RELA
SCHEMBL10042849 0.90 ACHE (0.47) ACHENPC1RAB9ATDP1RELA
SCHEMBL16449917 0.90 NPC1 (0.52) ACHENPC1RAB9ATDP1RELA
SCHEMBL14163840 0.90 NPC1 (0.52) ACHENPC1RAB9ATDP1RELA
SCHEMBL14570731 0.89 ACHE (0.48) APPACHENPC1RAB9ARELA
SCHEMBL13152209 0.89 ACHE (0.48) APPACHENPC1RAB9ARELA
SCHEMBL8944074 0.89 ACHE (0.48) ACHENPC1RAB9ATDP1RELA
SCHEMBL10065391 0.89 NPC1 (0.51) ACHENPC1RAB9ATDP1RELA
SCHEMBL10042851 0.86 ACHE (0.43) APPACHENPC1RAB9ATDP1
SCHEMBL17401210 0.86 MEN1 (0.53) APPACHENPC1RAB9ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1354887-B1 Ligands for metals and improved metal-catalyzed processes based thereon MASSACHUSETTS INST TECHNOLOGY (US) 2007-04-25 EP disclosed
EP-1097158-B1 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INST TECHNOLOGY (US) 2006-01-25 EP disclosed
EP-1097158-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2001-05-09 EP disclosed
WO-2000002887-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2000-01-20 WO disclosed