Guanidine

Guanidine

SCHEMBL5611641

CCOC(C(=O)O)C(O)C(O)C(O)CO.N=C(N)N

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2

The experimentally established mechanism targets of Guanidine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.44
SLCO1B1 Q9Y6L6 1/20 0.44
PDE4A P27815 1/20 0.43
LMNA P02545 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
KDM4E B2RXH2 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1133839 0.92 PDE4A (0.50) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL5173596 0.90 PDE4A (0.48) USP2SLCO1B1PDE4ALMNAL3MBTL1
Malonic Acid SCHEMBL17966082 0.85 PDE4A (0.44) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL6550889 0.78 PDE4A (0.42) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL3952432 0.78 PDE4A (0.42) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL6498093 0.77 PDE4A (0.46) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL5559507 0.75 LMNA (0.48) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL3899113 0.75 LMNA (0.48) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL11210752 0.75 LMNA (0.48) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL4734230 0.75 LMNA (0.53) USP2SLCO1B1PDE4ALMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1417064-A4 LUBRICANT SYSTEM FOR USE IN POWDERED METALS APEX ADVANCED TECHNOLOGIES LLC (US) 2006-12-20 EP claimed
US-20040175286-A1 Lubricant system for use in powdered metals APEX ADVANCED TECHNOLOGIES, LLC 2004-09-09 US claimed
EP-1417064-A1 LUBRICANT SYSTEM FOR USE IN POWDERED METALS Apex Advanced Technologies, LLC (US) 2004-05-12 EP claimed
US-20040077508-A1 Lubricant system for use in powdered metals APEX ADVANCED TECHNOLOGIES, LLC 2004-04-22 US claimed
US-6679935-B2 PRESSURIZING A SOLID LUBRICANT AND CONVERTING TO A LIQUID PHASE; USING IN MOLDING METAL POWDER OR PRESSING CERAMIC POWDER APEX ADVANCED TECHNOLOGIES, LLC 2004-01-20 US claimed
US-20030109388-A1 Lubricant system for use in powdered metals JOHNSON ELECTRIC NORTH AMERICA, INC. 2003-06-12 US claimed
WO-2003015962-A1 LUBRICANT SYSTEM FOR USE IN POWDERED METALS APEX ADVANCED TECHNOLOGIES, LLC (US) 2003-02-27 WO claimed
US-7264646-B2 Lubricant system for use in powdered metals APEX ADVANCED TECHNOLOGIES, LLC (US) 2007-09-04 US disclosed
EP-1417064-A4 LUBRICANT SYSTEM FOR USE IN POWDERED METALS APEX ADVANCED TECHNOLOGIES LLC (US) 2006-12-20 EP disclosed
US-20040175286-A1 Lubricant system for use in powdered metals APEX ADVANCED TECHNOLOGIES, LLC 2004-09-09 US disclosed
EP-1417064-A1 LUBRICANT SYSTEM FOR USE IN POWDERED METALS Apex Advanced Technologies, LLC (US) 2004-05-12 EP disclosed
US-20040077508-A1 Lubricant system for use in powdered metals APEX ADVANCED TECHNOLOGIES, LLC 2004-04-22 US disclosed
US-6679935-B2 PRESSURIZING A SOLID LUBRICANT AND CONVERTING TO A LIQUID PHASE; USING IN MOLDING METAL POWDER OR PRESSING CERAMIC POWDER APEX ADVANCED TECHNOLOGIES, LLC 2004-01-20 US disclosed
US-20030109388-A1 Lubricant system for use in powdered metals JOHNSON ELECTRIC NORTH AMERICA, INC. 2003-06-12 US disclosed
WO-2003015962-A1 LUBRICANT SYSTEM FOR USE IN POWDERED METALS APEX ADVANCED TECHNOLOGIES, LLC (US) 2003-02-27 WO disclosed