SCHEMBL5613755

SCHEMBL5613755

NC(=O)c1cnc2cc[nH]c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.46
HPGDS O60760 2/20 0.44
PIK3C3 Q8NEB9 1/20 0.44
RIPK1 Q13546 1/20 0.43
NNMT P40261 5/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
CCNT1 O60563 1/20 0.41
CCND1 P24385 1/20 0.41
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
CDK7 P50613 1/20 0.41
CDK9 P50750 1/20 0.41
CCNH P51946 1/20 0.41
MNAT1 P51948 1/20 0.41
CDK6 Q00534 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31508289 1.00 MAPK1 (0.46) MAPK1HPGDSPIK3C3RIPK1NNMT
SCHEMBL30569172 0.84 ALDH1A1 (0.51) PIK3C3SMN1; SMN2HDAC6KDM4EALDH1A1
SCHEMBL1607825 0.84 ALDH1A1 (0.51) PIK3C3SMN1; SMN2HDAC6KDM4EALDH1A1
SCHEMBL12709594 0.83 PIK3C3 (0.50) PIK3C3SMN1; SMN2CDK8CDK7HDAC6
SCHEMBL31194336 0.83 PIK3C3 (0.50) PIK3C3SMN1; SMN2CDK8CDK7HDAC6
SCHEMBL4145595 0.82 PIK3C3 (0.47) PIK3C3SMN1; SMN2HDAC6KDM4EALDH1A1
SCHEMBL1608350 0.80 HDAC6 (0.60) PIK3C3SMN1; SMN2HDAC6HTTAPP
SCHEMBL4410049 0.79 PIK3C3 (0.44) HPGDSPIK3C3SMN1; SMN2HDAC6KDM4E
SCHEMBL2671386 0.79 PIK3C3 (0.47) MAPK1PIK3C3CDK8HDAC6KDM4E
SCHEMBL20364680 0.79 PIK3C3 (0.44) PIK3C3SMN1; SMN2HDAC6KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023130054-A2 HETEROARYL COMPOUNDS AS INHIBITORS OF IRAK4, COMPOSITIONS AND APPLICATIONS THEREOF ACCRO BIOSCIENCE (HK) LIMITED (CN) 2023-07-06 WO disclosed
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed
EP-1784403-A1 PYRROLO[3,2-B]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF Yuhan Corporation (KR) 2007-05-16 EP disclosed
WO-2006038773-A1 PYRROLO[3,2-B]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2006-04-13 WO disclosed