SCHEMBL5614263

SCHEMBL5614263

COc1ccc(-c2cnc3nc([AsH]CCc4ccccc4)nc(N)c3n2)cc1OC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.57
MAPK1 P28482 3/20 0.42
GAK O14976 1/20 0.41
AGTR1 P30556 1/20 0.40
GSK3B P49841 1/20 0.40
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDE4A P27815 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
ADORA1 P30542 1/20 0.39
NEK2 P51955 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5461580 0.81 NOS1 (0.57) NOS1MAPK1AGTR1LMNAADORA1
SCHEMBL5614262 0.80 NOS1 (0.51) NOS1MAPK1GAKAGTR1L3MBTL1
SCHEMBL5456792 0.79 NOS1 (0.60) NOS1AGTR1ADORA1
SCHEMBL6064072 0.75 NOS1 (0.65) NOS1MAPK1KDM4EMEN1ALDH1A1
SCHEMBL4451753 0.73 NOS1 (0.53) NOS1GAKAGTR1PDE4BNEK2
SCHEMBL6063982 0.73 NOS1 (0.69) NOS1KDM4EALDH1A1HPGD
SCHEMBL5508808 0.73 NOS1 (1.00) NOS1MAPK1AGTR1ADORA1KDM4E
Water SCHEMBL6483834 0.72 NOS1 (0.98) NOS1MAPK1AGTR1ADORA1KDM4E
Water SCHEMBL6483831 0.72 NOS1 (0.98) NOS1MAPK1AGTR1ADORA1KDM4E
SCHEMBL5461575 0.72 NOS1 (0.51) NOS1MAPK1AGTR1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673092-B1 HETEROCYCLE-SUBSTITUTED PTERIDINE DERIVATIVES AND THEIR USE IN THERAPY 4 AZA IP NV (BE) 2007-08-15 EP disclosed