SCHEMBL561497

SCHEMBL561497

CCOC(=O)c1cc[nH]n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.56
TSHR P16473 1/20 0.47
PDE4D Q08499 1/20 0.46
KMT2A Q03164 2/20 0.46
KDM4E B2RXH2 4/20 0.45
MAPT P10636 3/20 0.45
NPSR1 Q6W5P4 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA7 P43166 2/20 0.44
CA9 Q16790 2/20 0.44
CA14 Q9ULX7 2/20 0.44
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
POLB P06746 3/20 0.44
NPC1 O15118 2/20 0.44
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Carbon Dioxide SCHEMBL28377710 0.95 CYP1A2 (0.51) CYP1A2TSHRPDE4DKMT2AKDM4E
SCHEMBL28125301 0.90 CYP1A2 (0.46) CYP1A2TSHRKMT2AKDM4EMAPT
SCHEMBL20488640 0.85 ALDH1A1 (0.50) CYP1A2TSHRKDM4EMAPTL3MBTL1
SCHEMBL29819645 0.85 CYP1A2 (0.43) CYP1A2TSHRPDE4DKMT2AKDM4E
SCHEMBL20570815 0.82 TSHR (0.53) CYP1A2TSHRPDE4DKDM4EMAPT
SCHEMBL21165934 0.81 CYP1A2 (0.41) CYP1A2TSHRPDE4DKMT2AKDM4E
SCHEMBL29291579 0.81 TSHR (0.54) CYP1A2TSHRPDE4DKDM4EMAPT
SCHEMBL27970370 0.81 TSHR (0.51) CYP1A2TSHRPDE4DKDM4EMAPT
SCHEMBL20357845 0.81 CYP1A2 (0.35) CYP1A2TSHRKMT2AKDM4EMAPT
SCHEMBL20920374 0.80 ALDH1A1 (0.51) CYP1A2TSHRKMT2AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1059 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110139862-B Substituted bicyclic heterocyclic derivatives useful as ROMK channel inhibitors 百时美施贵宝公司 2024-01-16 CN claimed
CN-113880769-B Chelating agent for metal zirconium marking and synthetic method and application thereof 华中科技大学 2023-03-31 CN claimed
CN-112107568-B Diaryl amide compound and application thereof 北京龙嘉博创医药科技有限公司 2022-03-25 CN claimed
CN-113880769-A Chelating agent for metal zirconium marking and synthetic method and application thereof 华中科技大学 2022-01-04 CN claimed
CN-212199075-U Impurity removing device for producing 4-pyrazole ethyl formate 南京麦瑞米生物技术有限公司 2020-12-22 CN claimed
CN-211799307-U Filter equipment is used in production of 4 pyrazole ethyl formate 南京麦瑞米生物技术有限公司 2020-10-30 CN claimed
CN-211800833-U Reation kettle is used in production of 4 pyrazole ethyl formate 南京麦瑞米生物技术有限公司 2020-10-30 CN claimed
CN-211771011-U 4 pyrazole ethyl formate purification device 南京麦瑞米生物技术有限公司 2020-10-27 CN claimed
CN-106187894-A The preparation method of 1 methyl 3 ethyl 4 chlorine 5 pyrazole carboxylic acid ethyl ester 潍坊鑫诺化工有限公司 2016-12-07 CN claimed
EP-2531490-A1 CYCLOHEXYL AMIDE DERIVATIVES AS CRF RECEPTOR ANTAGONISTS Novartis AG (CH) 2012-12-12 EP claimed
WO-2011095450-A1 CYCLOHEXYL AMIDE DERIVATIVES AS CRF RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2011-08-11 WO claimed
EP-1917247-A1 4,5-DIHYDR0-1H-PYRAZOLE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICAMENTS Laboratorios del Dr. Esteve S.A. (ES) 2008-05-07 EP claimed
WO-2007009690-A1 HETEROCYCLYL-SUBSTITUTED PYRAZOLINE COMPOUNDS, THEIR PREPARATION AND USE AS MEDICAMENTS LABORATORIOS DEL DR. ESTEVE, S.A (ES) 2007-01-25 WO claimed
WO-2007009689-A1 4,5-DIHYDR0-1H-PYRAZOLE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICAMENTS LABORATORIOS DEL DR.ESTEVE, S.A. (ES) 2007-01-25 WO claimed
CN-1449247-A Selective herbicides based on arylsulfonylaminocarbonyl triazolinones BAYER AG (DE) 2003-10-15 CN claimed
EP-0293220-B1 Pharmacologically active 2-and 3-substituted (1', 5'-diaryl-3-pyrazolyl)-N-Hydroxypropanamides and method for synthesizing ORTHO PHARMA CORP (US) 1994-08-31 EP claimed
EP-0293220-A2 Pharmacologically active 2-and 3-substituted (1', 5'-diaryl-3-pyrazolyl)-N-Hydroxypropanamides and method for synthesizing ORTHO PHARMACEUTICAL CORPORATION (US) 1988-11-30 EP claimed
JP-6041455-A None JP disclosed
JP-H0641455-A FIBER REACTIVE MONOAZO YELLOW DYE HOECHST CELANESE CORP 1994-02-15 JP disclosed
CN-86108643-A Insecticidal method using N-phenylpyrazoles 1987-07-29 CN disclosed