SCHEMBL5615411

SCHEMBL5615411

CC(C)(C)[C@H](O)C(=O)N[C@@H](C(Cc1ccc(-c2ccccn2)cc1)c1ccccc1)[C@@H](O)CCNC(=O)[C@@H](NC(=O)O)C(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UGT1A1 P22309 3/20 0.45
MLNR O43193 1/20 0.45
NR1I2 O75469 1/20 0.45
SLCO2B1 O94956 1/20 0.45
ABCB11 O95342 1/20 0.45
ABCB1 P08183 1/20 0.45
CCKAR P32238 1/20 0.45
OPRK1 P41145 1/20 0.45
GHSR Q92847 1/20 0.45
SLCO1B3 Q9NPD5 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
SLCO1B1 Q9Y6L6 1/20 0.45
CTSD P07339 2/20 0.39
CYP3A4 P08684 2/20 0.39
KCNH2 Q12809 1/20 0.39
CNR1 P21554 2/20 0.38
CNR2 P34972 1/20 0.38
TRPV1 Q8NER1 1/20 0.37
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4562736 0.83 UGT1A1 (0.44) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL6010546 0.81 CTSD (0.57) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL3812718 0.81 CTSD (0.54) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL6010531 0.81 UGT1A1 (0.43) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL6010283 0.81 UGT1A1 (0.43) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL5615281 0.80 CYP3A4 (0.56) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL5615413 0.80 CYP3A4 (0.56) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL5615374 0.80 CTSD (0.53) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL5615407 0.79 CYP3A4 (0.52) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL6010420 0.79 CTSD (0.60) UGT1A1MLNRNR1I2SLCO2B1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007516260-A 2007-06-21 JP claimed
EP-1697344-A2 HIV PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 2006-09-06 EP claimed
WO-2005058841-A2 HIV PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 2005-06-30 WO claimed