SCHEMBL5620132

SCHEMBL5620132

CCc1cc(C(N)=O)c2nc(C3CCCNC3)[nH]c2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.65
MAP4K4 O95819 2/20 0.48
INSR P06213 2/20 0.48
CSF1R P07333 2/20 0.48
PIM1 P11309 2/20 0.48
CLK2 P49760 2/20 0.48
IRAK1 P51617 2/20 0.48
MAP4K2 Q12851 2/20 0.48
DYRK1A Q13627 2/20 0.48
MINK1 Q8N4C8 2/20 0.48
AURKB Q96GD4 2/20 0.48
CLK4 Q9HAZ1 2/20 0.48
ALK Q9UM73 2/20 0.48
MAP4K5 Q9Y4K4 2/20 0.48
FLT4 P35916 1/20 0.48
FLT3 P36888 1/20 0.48
ITK Q08881 1/20 0.48
PIM3 Q86V86 1/20 0.48
HIPK2 Q9H2X6 1/20 0.48
MKNK2 Q9HBH9 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5620854 0.94 PARP1 (0.64) PARP1PARP2
SCHEMBL5621977 0.87 PARP1 (0.62) PARP1PARP2
SCHEMBL7040728 0.85 PARP1 (0.51) PARP1MAP4K4INSRCSF1RPIM1
SCHEMBL5622245 0.84 PARP1 (0.70) PARP1MAP4K4INSRCSF1RPIM1
SCHEMBL5620707 0.84 PARP1 (0.69) PARP1MAP4K4INSRCSF1RPIM1
SCHEMBL5620141 0.83 PARP1 (0.51) PARP1MAP4K4INSRCSF1RPIM1
SCHEMBL5621678 0.80 PARP1 (0.64) PARP1MAP4K4INSRCSF1RPIM1
SCHEMBL5621627 0.79 PARP1 (1.00) PARP1MAP4K4INSRCSF1RPIM1
SCHEMBL7043271 0.78 PARP1 (0.49) PARP1PARP2
Hydrochloric Acid SCHEMBL18614365 0.78 PARP1 (0.98) PARP1MAP4K4INSRCSF1RPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39608-E1 Substituted benzimidazoles and their use as PARP inhibitors ABBOTT GMBH & CO. KG (DE) 2007-05-01 US disclosed
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed