SCHEMBL7043271

SCHEMBL7043271

CCc1cc(OC(N)=O)c2nc(C3CCNC3)[nH]c2c1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.49
PARP2 Q9UGN5 2/20 0.38
HTR1F P30939 1/20 0.33
HTR2A P28223 1/20 0.33
BAZ2A Q9UIF9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7040728 0.94 PARP1 (0.51) PARP1PARP2HTR2ABAZ2A
SCHEMBL7046800 0.94 PARP1 (0.47) PARP1PARP2
SCHEMBL7045124 0.85 PARP1 (0.53) PARP1PARP2
SCHEMBL7040921 0.84 PARP1 (0.52) PARP1PARP2
SCHEMBL5620854 0.84 PARP1 (0.64) PARP1PARP2
SCHEMBL7042400 0.80 PARP1 (0.47) PARP1PARP2
SCHEMBL6869625 0.79 PARP1 (0.69) PARP1PARP2
SCHEMBL7411360 0.79 PARP1 (0.56) PARP1PARP2
SCHEMBL7042529 0.79 PARP1 (0.54) PARP1PARP2
SCHEMBL7038859 0.78 PARP1 (0.51) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed