SCHEMBL5624732

SCHEMBL5624732

O=C1NC(c2ccccc2)Oc2ccccc21

nearest known ligand 0.77

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.77
KMT2A Q03164 3/20 0.77
POLB P06746 1/20 0.77
KDM4E B2RXH2 7/20 0.65
HSD17B10 Q99714 5/20 0.65
ALDH1A1 P00352 4/20 0.65
USP2 O75604 1/20 0.65
GAA P10253 1/20 0.65
HPGD P15428 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7672741 0.81 MEN1 (0.50) MEN1KMT2APOLBKDM4EHSD17B10
SCHEMBL15678813 0.80 KDM4E (0.79) MEN1KMT2APOLBKDM4EHSD17B10
SCHEMBL14478875 0.80 KDM4E (1.00) MEN1KMT2APOLBKDM4EHSD17B10
SCHEMBL13402249 0.79 KDM4E (1.00) MEN1KMT2APOLBKDM4EHSD17B10
SCHEMBL12691232 0.77 KDM4E (0.59) MEN1KMT2APOLBKDM4EHSD17B10
SCHEMBL18324078 0.76 TNKS2 (0.52) MEN1KMT2APOLBKDM4EHSD17B10
SCHEMBL5626972 0.74 PARP1 (0.56) MEN1KMT2APOLBKDM4EHSD17B10
SCHEMBL541947 0.73 MEN1 (0.49) MEN1KMT2APOLBKDM4EHSD17B10
SCHEMBL30209785 0.73 MEN1 (0.49) MEN1KMT2APOLBKDM4EHSD17B10
SCHEMBL23175219 0.71 PARP1 (0.57) MEN1KMT2APOLBKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108774189-B Oxazine phenyl ether derivative and preparation method thereof 安徽师范大学 2022-04-19 CN claimed
US-20040043987-A1 Novel compounds and their use as positive AMPA receptor modulators NEUROSEARCH A/S. 2004-03-04 US claimed
CN-1293665-A New compounds and their use as positive AMPA receptor modulators NEUROSEARCH AS (DK) 2001-05-02 CN claimed
EP-1071426-A2 NOVEL COMPOUNDS AND THEIR USE AS POSITIVE AMPA RECEPTOR MODULATORS NEUROSEARCH A/S (DK) 2001-01-31 EP claimed
WO-1999042456-A2 NOVEL COMPOUNDS AND THEIR USE AS POSITIVE AMPA RECEPTOR MODULATORS NEUROSEARCH A/S (DK) 1999-08-26 WO claimed
CN-108774189-B Oxazine phenyl ether derivative and preparation method thereof 安徽师范大学 2022-04-19 CN disclosed
US-7235548-B2 Compounds and their use as positive AMPA receptor modulators NEUROSEARCH A/S (DK) 2007-06-26 US disclosed
US-6943159-B1 Compounds and their use as positive AMPA receptor modulators NEUROSEARCH A/S (DK) 2005-09-13 US disclosed
US-20040043987-A1 Novel compounds and their use as positive AMPA receptor modulators NEUROSEARCH A/S. 2004-03-04 US disclosed
CN-1293665-A New compounds and their use as positive AMPA receptor modulators NEUROSEARCH AS (DK) 2001-05-02 CN disclosed
EP-1071426-A2 NOVEL COMPOUNDS AND THEIR USE AS POSITIVE AMPA RECEPTOR MODULATORS NEUROSEARCH A/S (DK) 2001-01-31 EP disclosed
WO-1999042456-A2 NOVEL COMPOUNDS AND THEIR USE AS POSITIVE AMPA RECEPTOR MODULATORS NEUROSEARCH A/S (DK) 1999-08-26 WO disclosed
EP-0566018-B1 Benzoxazinone and benzothiazinone derivatives endowed with cardiovascular activity ITALFARMACO SPA (IT) 1998-08-05 EP disclosed
US-5480882-A Benzoxazinone and benzothiazinone derivatives having cardiovascular activity ITALFARMACO S.P.A. (IT) 1996-01-02 US disclosed
EP-0490183-B1 Benzoxazinone and benzothiazinone derivatives endowed with cardiovascular activity ITALFARMACO SPA (IT) 1995-04-19 EP disclosed
EP-0566018-A2 Benzoxazinone and benzothiazinone derivatives endowed with cardiovascular activity ITALFARMACO S.p.A. (IT) 1993-10-20 EP disclosed
US-5189034-A Vasodilating, antianginal agents ITALFARMACO S.P.A. (IT) 1993-02-23 US disclosed
EP-0490183-A1 Benzoxazinone and benzothiazinone derivatives endowed with cardiovascular activity ITALFARMACO S.p.A. (IT) 1992-06-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040043987-A1 Novel compounds and their use as positive AMPA receptor modulators GRIK4, GRIA4, GRM2 MEN1 4649/4885KMT2A 869/4885POLB 3401/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.