SCHEMBL5628554

SCHEMBL5628554

CC(=O)OCC1(c2cccc(C(F)(F)F)c2)CCNCC1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 9/20 0.56
SLC6A4 P31645 9/20 0.49
CCR2 P41597 1/20 0.46
SLC6A3 Q01959 2/20 0.45
SLC6A2 P23975 1/20 0.45
KCNH2 Q12809 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4813147 0.83 TACR1 (0.53) TACR1SLC6A4CCR2SLC6A3SLC6A2
SCHEMBL27607905 0.81 TACR1 (0.50) TACR1SLC6A4CCR2SLC6A3SLC6A2
SCHEMBL4631291 0.81 TACR1 (0.56) TACR1SLC6A4KCNH2
SCHEMBL4816350 0.80 TACR1 (0.48) TACR1SLC6A4SLC6A3SLC6A2
SCHEMBL6266690 0.79 SLC6A4 (0.51) TACR1SLC6A4CCR2SLC6A3SLC6A2
Hydrochloric Acid SCHEMBL27626949 0.78 CCR2 (0.46) TACR1SLC6A4CCR2SLC6A3SLC6A2
SCHEMBL8886072 0.77 CCR2 (0.45) TACR1SLC6A4CCR2SLC6A3SLC6A2
SCHEMBL2811089 0.77 TACR1 (0.53) TACR1SLC6A4CCR2SLC6A3SLC6A2
SCHEMBL12585395 0.77 SLC6A4 (0.74) TACR1SLC6A4SLC6A3SLC6A2KCNH2
SCHEMBL4848259 0.77 SLC6A4 (0.52) TACR1SLC6A4CCR2SLC6A3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7294628-B2 Piperazinylacylpiperidine derivatives, their preparation and therapeutic use thereof SANOFI-AVENTIS (FR) 2007-11-13 US disclosed