SCHEMBL5634535

SCHEMBL5634535

O=C(O)c1cccc(Oc2ccc(-c3nc4ccccc4[nH]3)cc2)c1

nearest known ligand 0.76

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 13/20 0.76
KDM4E B2RXH2 2/20 0.69
ALDH1A1 P00352 2/20 0.69
HPGD P15428 2/20 0.69
NPC1 O15118 1/20 0.69
RAB9A P51151 1/20 0.69
SMN1; SMN2 Q16637 1/20 0.69
KMT2A Q03164 1/20 0.64
DHODH Q02127 1/20 0.60
AKR1C3 P42330 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3925984 0.91 CHEK2 (0.74) CHEK2KDM4EALDH1A1HPGDNPC1
SCHEMBL2318980 0.86 CHEK2 (1.00) CHEK2
SCHEMBL3926681 0.86 CHEK2 (0.81) CHEK2KDM4EALDH1A1HPGDNPC1
SCHEMBL3918418 0.85 CHEK2 (0.84) CHEK2KMT2A
SCHEMBL6643299 0.85 CHEK2 (1.00) CHEK2KMT2A
SCHEMBL5252669 0.85 CHEK2 (0.70) CHEK2KDM4EALDH1A1HPGDNPC1
SCHEMBL3335320 0.84 KDM4E (0.71) CHEK2KDM4EALDH1A1HPGDNPC1
SCHEMBL3918297 0.84 CHEK2 (0.78) CHEK2KDM4EALDH1A1HPGDNPC1
SCHEMBL3927854 0.82 CHEK2 (0.71) CHEK2KDM4EALDH1A1HPGDNPC1
SCHEMBL31679082 0.82 KDM4E (1.00) CHEK2KDM4EALDH1A1HPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7271261-B2 Substituted benzimidazoles and imidazo-[4,5]-pyridines ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2007-09-18 US claimed
US-7271261-B2 Substituted benzimidazoles and imidazo-[4,5]-pyridines ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2007-09-18 US disclosed