SCHEMBL5635111

SCHEMBL5635111

Cc1cc(F)ccc1Nc1cc2c3c(c1)[C@@H]1CNCC[C@@H]1N3CCCS2

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 18/20 0.58
HTR2A P28223 15/20 0.54
HTR2B P41595 3/20 0.54
DRD2 P14416 13/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5636311 0.88 HTR2C (0.52) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636500 0.87 HTR2C (0.64) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637649 0.84 HTR2C (0.58) HTR2CHTR2AHTR2BDRD2
SCHEMBL6490555 0.83 HTR2C (0.40) HTR2CHTR2AHTR2B
SCHEMBL5638318 0.83 HTR2C (0.69) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636092 0.82 HTR2C (0.56) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636264 0.81 HTR2C (0.65) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637044 0.81 HTR2C (0.69) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636844 0.80 HTR2C (0.72) HTR2CHTR2AHTR2BDRD2
SCHEMBL6502139 0.79 HTR2C (0.36) HTR2CHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed