SCHEMBL5636092

SCHEMBL5636092

Clc1ccc(Nc2cc3c4c(c2)[C@@H]2CNCC[C@@H]2N4CCCS3)c(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.56
HTR2A P28223 6/20 0.56
HTR2B P41595 2/20 0.56
DRD2 P14416 4/20 0.37
JAK3 P52333 1/20 0.36
DPP4 P27487 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5636264 0.83 HTR2C (0.65) HTR2CHTR2AHTR2BDRD2
SCHEMBL6501819 0.83 HTR2C (0.38) HTR2CHTR2AHTR2BJAK3DPP4
SCHEMBL6502084 0.83 HTR2C (0.38) HTR2CHTR2AHTR2BJAK3DPP4
SCHEMBL5636247 0.82 HTR2C (0.76) HTR2CHTR2AHTR2BDRD2
SCHEMBL255569 0.82 HTR2C (0.76) HTR2CHTR2AHTR2BDRD2
SCHEMBL5635111 0.82 HTR2C (0.58) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636500 0.81 HTR2C (0.64) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636311 0.81 HTR2C (0.52) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636191 0.80 HTR2C (0.66) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637649 0.80 HTR2C (0.58) HTR2CHTR2AHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed