SCHEMBL5635151

SCHEMBL5635151

CCOc1ccc(-c2cc3c4c(c2)[C@@H]2CNCC[C@@H]2N4CCCO3)c(C(F)(F)F)c1

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 8/20 0.62
HTR2C P28335 6/20 0.62
HTR2B P41595 3/20 0.62
ACP1 P24666 1/20 0.33
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5637157 0.95 HTR2A (0.59) HTR2AHTR2CHTR2BACP1
SCHEMBL5636468 0.91 HTR2C (0.75) HTR2AHTR2CHTR2B
SCHEMBL15800579 0.89 HTR2C (0.62) HTR2AHTR2CHTR2B
SCHEMBL5636371 0.89 HTR2C (0.62) HTR2AHTR2CHTR2B
SCHEMBL29388613 0.89 HTR2C (0.62) HTR2AHTR2CHTR2B
SCHEMBL5635413 0.88 HTR2C (0.60) HTR2AHTR2CHTR2B
SCHEMBL5413061 0.86 HTR2C (0.83) HTR2AHTR2CHTR2BACP1
SCHEMBL5636686 0.86 HTR2C (0.72) HTR2AHTR2CHTR2B
SCHEMBL5638490 0.85 HTR2C (0.56) HTR2AHTR2CHTR2B
SCHEMBL5637064 0.85 HTR2C (0.56) HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed