SCHEMBL5635170

SCHEMBL5635170

FC(F)(F)c1ccc(-c2cc3c4c(c2)[C@@H]2CNCC[C@@H]2N4CCO3)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 6/20 0.46
HTR2A P28223 4/20 0.46
HTR2B P41595 4/20 0.46
AKT1 P31749 2/20 0.33
HTR6 P50406 1/20 0.32
PLAT P00750 2/20 0.32
SCN9A Q15858 1/20 0.32
TNIK Q9UKE5 1/20 0.31
TMEM97 Q5BJF2 1/20 0.31
KCNH2 Q12809 1/20 0.31
ROCK2 O75116 1/20 0.30
ROCK1 Q13464 1/20 0.30
ACP1 P24666 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5638182 0.95 HTR2C (0.48) HTR2CHTR2AHTR2BAKT1HTR6
SCHEMBL5637734 0.90 HTR2C (0.54) HTR2CHTR2AHTR2BHTR6PLAT
SCHEMBL5637209 0.88 HTR2C (0.42) HTR2CHTR2AHTR2BAKT1
SCHEMBL5636639 0.88 HTR2C (0.48) HTR2CHTR2AHTR2BAKT1HTR6
SCHEMBL5638389 0.87 HTR2C (0.43) HTR2CHTR2AHTR2BHTR6TNIK
SCHEMBL5410508 0.84 HTR2C (0.58) HTR2CHTR2AHTR2BPLATKCNH2
SCHEMBL5410506 0.84 HTR2C (0.58) HTR2CHTR2AHTR2BPLATKCNH2
SCHEMBL5636624 0.84 HTR2C (0.53) HTR2CHTR2AHTR2BHTR6TNIK
SCHEMBL5410691 0.83 HTR2C (0.66) HTR2CHTR2AHTR2BKCNH2ACP1
SCHEMBL5410687 0.83 HTR2C (0.66) HTR2CHTR2AHTR2BKCNH2ACP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed