SCHEMBL5638182

SCHEMBL5638182

FC(F)(F)c1ccc(-c2cc3c4c(c2)[C@@H]2CNCC[C@@H]2N4CCCO3)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 6/20 0.48
HTR2A P28223 5/20 0.48
HTR2B P41595 4/20 0.48
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ACP1 P24666 1/20 0.33
KCNH2 Q12809 1/20 0.32
HTR6 P50406 1/20 0.31
PLAT P00750 2/20 0.31
AKT1 P31749 2/20 0.30
CTSV O60911 1/20 0.30
CTSL P07711 1/20 0.30
CTSB P07858 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5635170 0.95 HTR2C (0.46) HTR2CHTR2AHTR2BACP1KCNH2
SCHEMBL5636451 0.88 HTR2C (0.51) HTR2CHTR2AHTR2BKMT2AALDH1A1
SCHEMBL5636401 0.85 HTR2C (0.45) HTR2CHTR2AHTR2BKCNH2HTR6
SCHEMBL5410687 0.85 HTR2C (0.66) HTR2CHTR2AHTR2BKMT2AMEN1
SCHEMBL5410691 0.85 HTR2C (0.66) HTR2CHTR2AHTR2BKMT2AMEN1
SCHEMBL5637734 0.85 HTR2C (0.54) HTR2CHTR2AHTR2BKMT2AMEN1
SCHEMBL5636687 0.84 HTR2C (0.56) HTR2CHTR2AHTR2BHTR6
SCHEMBL5405461 0.84 HTR2C (0.62) HTR2CHTR2AHTR2BKMT2AMEN1
SCHEMBL5637170 0.83 HTR2C (0.54) HTR2CHTR2AHTR2BKCNH2CYP2D6
SCHEMBL5636424 0.83 HTR2C (0.47) HTR2CHTR2AHTR2BACP1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed