SCHEMBL5635201

SCHEMBL5635201

COc1ccc(-c2cc3c4c(c2)C2CCNCCC2N4CCCS3)c(C)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 9/20 0.53
HTR2B P41595 5/20 0.49
HTR2A P28223 4/20 0.49
HTR3E A5X5Y0 1/20 0.35
HTR3B O95264 1/20 0.35
HTR3A P46098 1/20 0.35
HTR3D Q70Z44 1/20 0.35
HTR3C Q8WXA8 1/20 0.35
RYR2 Q92736 3/20 0.34
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33
KCNH2 Q12809 1/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.31
MCHR1 Q99705 1/20 0.31
PLAT P00750 1/20 0.31
HSD11B1 P28845 1/20 0.30
DRD2 P14416 1/20 0.30
JAK2 O60674 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5638466 0.94 HTR2C (0.61) HTR2CHTR2BHTR2AHTR3EHTR3B
SCHEMBL5637994 0.90 HTR2C (0.54) HTR2CHTR2BHTR2AHTR3ARYR2
Hydrochloric Acid SCHEMBL5637631 0.88 HTR2C (0.54) HTR2CHTR2BHTR2AHTR3EHTR3B
SCHEMBL5636958 0.85 HTR2C (0.62) HTR2CHTR2BHTR2ARYR2KCNH2
SCHEMBL5636853 0.84 HTR2C (0.59) HTR2CHTR2BHTR2AKDM4EALDH1A1
SCHEMBL5636633 0.84 HTR2C (0.61) HTR2CHTR2BHTR2ARYR2KCNH2
SCHEMBL5636700 0.84 HTR2C (0.68) HTR2CHTR2BHTR2AALDH1A1DRD2
SCHEMBL5637149 0.82 HTR2C (0.59) HTR2CHTR2BHTR2ARYR2DRD2
SCHEMBL5638149 0.82 HTR2C (0.66) HTR2CHTR2BHTR2ADRD2
SCHEMBL5636095 0.82 HTR2C (0.58) HTR2CHTR2BHTR2ARYR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed