SCHEMBL5635971

SCHEMBL5635971

CC(C)(C)OC(=O)N1CC[C@H]2[C@@H](C1)c1cc(-c3c(Cl)cccc3Cl)cc3c1N2CCO3

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 3/20 0.47
MAPT P10636 2/20 0.42
STS P08842 4/20 0.40
HTR2A P28223 5/20 0.39
HTR2C P28335 5/20 0.39
DRD2 P14416 4/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CNR1 P21554 1/20 0.37
HTR1A P08908 1/20 0.37
DRD4 P21917 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
TP53 P04637 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5637776 0.91 USP30 (0.49) USP30MAPTSTSHTR2AHTR2C
SCHEMBL5636680 0.86 USP30 (0.43) USP30MAPTSTSMEN1KMT2A
SCHEMBL5637027 0.86 USP30 (0.46) USP30MAPTSTSMEN1KMT2A
SCHEMBL5635159 0.85 USP30 (0.42) USP30MAPTHTR2AHTR2CDRD2
SCHEMBL5636646 0.84 USP30 (0.47) USP30MAPTHTR2AHTR2CDRD2
SCHEMBL5848904 0.83 STS (0.41) USP30MAPTSTSHTR2AHTR2C
SCHEMBL5636142 0.83 USP30 (0.44) USP30MAPTCNR1TP53LMNA
SCHEMBL5849542 0.83 STS (0.40) USP30MAPTSTSHTR2AHTR2C
SCHEMBL5636694 0.82 USP30 (0.53) USP30MAPT
SCHEMBL5636262 0.82 CNR1 (0.41) USP30MAPTSTSHTR2CMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed