SCHEMBL5636142

SCHEMBL5636142

CC(C)(C)OC(=O)N1CC[C@H]2[C@@H](C1)c1cc(-c3ccc(Cl)c(Cl)c3)cc3c1N2CCCO3

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 5/20 0.44
PTPN2 P17706 1/20 0.37
PTPN1 P18031 1/20 0.37
PTPN6 P29350 1/20 0.37
OPRK1 P41145 1/20 0.37
MAPT P10636 1/20 0.36
NTRK1 P04629 1/20 0.36
KAT6A Q92794 1/20 0.36
KAT5 Q92993 1/20 0.36
PARP1 P09874 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
CNR1 P21554 1/20 0.35
TP53 P04637 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5636828 0.89 USP30 (0.40) USP30MAPTCNR1TP53LMNA
SCHEMBL5636694 0.88 USP30 (0.53) USP30MAPT
SCHEMBL5637027 0.88 USP30 (0.46) USP30MAPTPARP1PARP2CNR1
SCHEMBL5636405 0.88 PIK3CD (0.46) USP30PDE4APDE4BPDE4C
SCHEMBL5636262 0.87 CNR1 (0.41) USP30MAPTCNR1TP53ALDH1A1
SCHEMBL5636680 0.86 USP30 (0.43) USP30MAPTCNR1TP53LMNA
SCHEMBL5636040 0.86 USP30 (0.46) USP30MAPTKAT6AKAT5TP53
SCHEMBL5846974 0.85 NPC1 (0.40) USP30PTPN2PTPN1PTPN6OPRK1
SCHEMBL5636737 0.85 USP30 (0.38) USP30MAPTTP53PDE4BALDH1A1
SCHEMBL5848258 0.85 NPC1 (0.40) USP30PTPN2PTPN1PTPN6OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed