SCHEMBL5635995

SCHEMBL5635995

CCOc1ccc(-c2cc3c4c(c2)[C@@H]2CNCC[C@@H]2N4CCCS3)c(Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.58
HTR2A P28223 6/20 0.52
HTR2B P41595 2/20 0.52
DRD2 P14416 2/20 0.32
ERN1 O75460 1/20 0.32
MCHR1 Q99705 1/20 0.32
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
POLB P06746 1/20 0.30
EIF4E P06730 1/20 0.30
KDM4E B2RXH2 1/20 0.30
USP2 O75604 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
TSHR P16473 1/20 0.30
HSD17B10 Q99714 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5636853 0.91 HTR2C (0.59) HTR2CHTR2AHTR2BDRD2MAOA
SCHEMBL5636633 0.91 HTR2C (0.61) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636297 0.88 HTR2C (0.58) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637619 0.88 HTR2A (0.62) HTR2CHTR2AHTR2BDRD2
SCHEMBL5638586 0.87 HTR2C (0.61) HTR2CHTR2AHTR2BDRD2
SCHEMBL5638412 0.87 HTR2C (0.61) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637189 0.86 HTR2C (0.64) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636247 0.86 HTR2C (0.76) HTR2CHTR2AHTR2BDRD2
SCHEMBL255569 0.86 HTR2C (0.76) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637994 0.84 HTR2C (0.54) HTR2CHTR2AHTR2BDRD2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed