SCHEMBL5638586

SCHEMBL5638586

FC(F)(F)Oc1ccc(-c2cc3c4c(c2)[C@H]2CNCC[C@H]2N4CCCS3)c(Cl)c1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.61
HTR2A P28223 3/20 0.52
HTR2B P41595 2/20 0.52
DRD2 P14416 1/20 0.31
TACR1 P25103 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5638412 0.90 HTR2C (0.61) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636633 0.90 HTR2C (0.61) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636185 0.89 HTR2C (0.66) HTR2CHTR2AHTR2BDRD2TACR1
SCHEMBL5637184 0.88 HTR2C (0.63) HTR2CHTR2AHTR2BDRD2
SCHEMBL5635995 0.87 HTR2C (0.58) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636297 0.87 HTR2C (0.58) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637598 0.87 HTR2C (0.69) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636247 0.87 HTR2C (0.76) HTR2CHTR2AHTR2BDRD2
SCHEMBL255569 0.87 HTR2C (0.76) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636778 0.85 HTR2C (0.67) HTR2CHTR2AHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed