SCHEMBL5636374

SCHEMBL5636374

FC(F)(F)c1ccc2c3c1c1c(n3CCS2)CCNC1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.36
HTR2A P28223 5/20 0.36
HTR2B P41595 1/20 0.36
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
TP53 P04637 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
ALOX15 P16050 1/20 0.31
MAPK1 P28482 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
LIPG Q9Y5X9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6486605 0.91 HTR2C (0.36) HTR2CHTR2AHTR2BLIPG
SCHEMBL5638608 0.78 HTR2C (0.50) HTR2CHTR2AKDM4EMEN1TP53
SCHEMBL11427742 0.77 HTR2C (0.47) HTR2CHTR2AKDM4EMEN1TP53
SCHEMBL6485539 0.76 HTR2C (0.47) HTR2CHTR2AHTR2B
Hydrochloric Acid SCHEMBL5636963 0.76 HTR2C (0.46) HTR2CHTR2AKDM4EMEN1TP53
SCHEMBL5636929 0.76 HTR2C (0.37) HTR2CHTR2AKDM4EMEN1TP53
SCHEMBL5635522 0.76 HTR2C (0.34) HTR2CHTR2AHTR2BKDM4EMEN1
SCHEMBL5637197 0.74 HTR2C (0.32) HTR2C
SCHEMBL6497657 0.73 HTR2C (0.38) HTR2CHTR2AHTR2B
SCHEMBL6483124 0.73 HTR2C (0.38) HTR2CHTR2AKDM4EMEN1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed