SCHEMBL5636581

SCHEMBL5636581

CC(C)(C)OC(=O)N1CC[C@H]2[C@@H](C1)c1cc(-c3ccc(F)cc3Cl)cc3c1N2CCCS3

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 15/20 0.45
DRD2 P14416 13/20 0.42
HTR2A P28223 13/20 0.42
NTRK1 P04629 2/20 0.39
PAK1 Q13153 1/20 0.38
TACR3 P29371 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5634987 0.92 HTR2C (0.54) HTR2CDRD2HTR2APAK1
SCHEMBL5636180 0.92 HTR2C (0.54) HTR2CDRD2HTR2APAK1
SCHEMBL5636957 0.89 HTR2C (0.43) HTR2CDRD2HTR2A
SCHEMBL5636141 0.89 HTR2C (0.50) HTR2CDRD2HTR2A
SCHEMBL5636395 0.88 HTR2C (0.43) HTR2CDRD2HTR2A
SCHEMBL5637659 0.88 HTR2C (0.48) HTR2CDRD2HTR2APAK1
SCHEMBL5638128 0.86 HTR2C (0.55) HTR2CDRD2HTR2A
SCHEMBL5637526 0.86 HTR2C (0.55) HTR2CDRD2HTR2A
SCHEMBL5638331 0.86 HTR2C (0.41) HTR2CDRD2HTR2APAK1
SCHEMBL5635470 0.85 HTR2C (0.47) HTR2CDRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed