SCHEMBL5634987

SCHEMBL5634987

CC(C)(C)OC(=O)N1CCC2C(C1)c1cc(-c3ccc(Cl)cc3Cl)cc3c1N2CCCS3

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 12/20 0.54
DRD2 P14416 10/20 0.44
HTR2A P28223 10/20 0.44
CNR1 P21554 3/20 0.39
CNR2 P34972 2/20 0.37
PAK1 Q13153 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
ALDH1A1 P00352 1/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5636180 1.00 HTR2C (0.54) HTR2CDRD2HTR2ACNR1CNR2
SCHEMBL5637659 0.96 HTR2C (0.48) HTR2CDRD2HTR2ACNR1CNR2
SCHEMBL5637526 0.94 HTR2C (0.55) HTR2CDRD2HTR2ACNR1CNR2
SCHEMBL5638128 0.94 HTR2C (0.55) HTR2CDRD2HTR2ACNR1CNR2
SCHEMBL5636581 0.92 HTR2C (0.45) HTR2CDRD2HTR2APAK1
SCHEMBL5636957 0.90 HTR2C (0.43) HTR2CDRD2HTR2A
SCHEMBL5636395 0.89 HTR2C (0.43) HTR2CDRD2HTR2AMAPTALDH1A1
SCHEMBL5638054 0.87 HTR2C (0.47) HTR2CDRD2HTR2AMAPT
SCHEMBL5635470 0.87 HTR2C (0.47) HTR2CDRD2HTR2AMAPT
SCHEMBL5848567 0.86 HTR2C (0.41) HTR2CHTR2ACNR1CNR2PAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed