SCHEMBL5637552

SCHEMBL5637552

COC(=O)/C=C\c1cc(OC)ccc1-c1cc2c3c(c1)[C@@H]1CNCC[C@@H]1N3CCCS2

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 13/20 0.53
HTR2A P28223 8/20 0.49
HTR2B P41595 5/20 0.49
L3MBTL1 Q9Y468 1/20 0.34
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
HTT P42858 1/20 0.32
DRD2 P14416 5/20 0.32
RYR2 Q92736 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5636295 1.00 HTR2C (0.53) HTR2CHTR2AHTR2BL3MBTL1KDM4E
SCHEMBL6756313 0.93 HTR2C (0.53) HTR2CHTR2AHTR2BL3MBTL1KDM4E
SCHEMBL5636494 0.88 HTR2C (0.58) HTR2CHTR2AHTR2BDRD2RYR2
SCHEMBL5637051 0.88 HTR2C (0.54) HTR2CHTR2AHTR2B
SCHEMBL5636533 0.88 HTR2C (0.54) HTR2CHTR2AHTR2B
SCHEMBL5636382 0.87 HTR2C (0.37) HTR2CHTR2AHTR2BL3MBTL1DRD2
SCHEMBL5636083 0.87 HTR2C (0.37) HTR2CHTR2AHTR2BL3MBTL1DRD2
SCHEMBL5636128 0.86 HTR2C (0.57) HTR2CHTR2AHTR2BKDM4EDRD2
SCHEMBL5636580 0.85 HTR2C (0.58) HTR2CHTR2AHTR2BDRD2RYR2
SCHEMBL5636958 0.84 HTR2C (0.62) HTR2CHTR2AHTR2BKMT2ARYR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed