SCHEMBL5638522

SCHEMBL5638522

Fc1cccc(-c2cc3c4c(c2)[C@@H]2CNCC[C@@H]2N4CCS3)c1F

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 13/20 0.74
HTR2A P28223 10/20 0.55
HTR2B P41595 3/20 0.55
DRD2 P14416 7/20 0.34
WNT1 P04628 1/20 0.32
DYRK1A Q13627 1/20 0.32
CHEK1 O14757 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5636715 0.89 HTR2C (0.88) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637548 0.86 HTR2C (0.74) HTR2CHTR2AHTR2BDRD2
SCHEMBL5638100 0.85 HTR2C (1.00) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636712 0.85 HTR2C (1.00) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636530 0.84 HTR2C (0.62) HTR2CHTR2AHTR2BDRD2
Hydrochloric Acid SCHEMBL6754234 0.83 HTR2C (0.79) HTR2CHTR2AHTR2BDRD2
SCHEMBL5415873 0.82 HTR2C (0.60) HTR2CHTR2AHTR2BDRD2WNT1
SCHEMBL5636052 0.81 HTR2C (0.52) HTR2CHTR2AHTR2BDRD2WNT1
SCHEMBL5410641 0.81 HTR2C (0.56) HTR2CHTR2AHTR2BDRD2WNT1
SCHEMBL5637517 0.80 HTR2C (0.89) HTR2CHTR2AHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed