SCHEMBL564135

SCHEMBL564135

Brc1c(NC2NCCN2)ccc2nccnc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 14/20 0.55
ADRA2C P18825 13/20 0.55
ADRA2B P18089 12/20 0.55
ADRA1D P25100 11/20 0.55
ADRA1A P35348 9/20 0.55
ADRA1B P35368 8/20 0.55
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 2/20 0.55
MAPT P10636 2/20 0.55
NR1I2 O75469 1/20 0.55
LMNA P02545 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
HTR1A P08908 1/20 0.55
CYP2D6 P10635 1/20 0.55
HPGD P15428 1/20 0.55
ALOX15 P16050 1/20 0.55
MAPK1 P28482 1/20 0.55
BLM P54132 1/20 0.55
HSD17B10 Q99714 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9341170 0.98 ADRA2A (0.53) ADRA2AADRA2CADRA2BADRA1DADRA1A
SCHEMBL8153481 0.82 ADRA2A (0.55) ADRA2AADRA2CADRA2BADRA1DADRA1A
SCHEMBL7202916 0.74 RIPK2 (0.33)
Brimonidine SCHEMBL24670 0.71 ADRA2A (1.00) ADRA2AADRA2CADRA2BADRA1DADRA1A
SCHEMBL22224522 0.71 ADRA2A (0.59) ADRA2AADRA2CADRA2BADRA1DADRA1A
Brimonidine SCHEMBL20511531 0.71 ADRA2A (1.00) ADRA2AADRA2CADRA2BADRA1DADRA1A
Brimonidine SCHEMBL29374525 0.71 ADRA2A (1.00) ADRA2AADRA2CADRA2BADRA1DADRA1A
Brimonidine SCHEMBL22616115 0.70 ADRA2A (0.97) ADRA2AADRA2CADRA2BADRA1DADRA1A
Brimonidine SCHEMBL1685506 0.70 ADRA2A (0.97) ADRA2AADRA2CADRA2BADRA1DADRA1A
SCHEMBL22172211 0.69 ADRA2A (0.51) ADRA2AADRA2CADRA2BADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0537165-B1 POLYMERIC DRUG DELIVERY SYSTEM ALLERGAN INC (US) 1998-07-01 EP claimed
US-5474780-A Monolithic maleic anhydride drug delivery systems ALLERGAN, INC. (US) 1995-12-12 US claimed
EP-0630262-A1 COMPOSITIONS FOR CONTROLLED DELIVERY OF PHARMACEUTICAL COMPOUNDS ALLERGAN, INC. (US) 1994-12-28 EP claimed
US-5275820-A Stable suspension formulations of bioerodible polymer matrix microparticles incorporating drug loaded ion exchange resin particles ALLERGAN, INC. (US) 1994-01-04 US claimed
EP-0564537-A1 STABLE SUSPENSION FORMULATIONS FOR CONTROLLED DELIVERY OF PHARMACEUTICAL COMPOUNDS ALLERGAN, INC. (US) 1993-10-13 EP claimed
WO-1993017716-A1 COMPOSITIONS FOR CONTROLLED DELIVERY OF PHARMACEUTICAL COMPOUNDS ALLERGAN, INC. (US) 1993-09-16 WO claimed
US-5215991-A Administering amiloride and an imidazolidine derivative ALLERGAN, INC. (US) 1993-06-01 US claimed
EP-0537165-A1 POLYMERIC DRUG DELIVERY SYSTEM ALLERGAN, INC. (US) 1993-04-21 EP claimed
EP-0537165-A4 POLYMERIC DRUG DELIVERY SYSTEM. ALLERGAN INC (US) 1993-02-24 EP claimed
US-5180721-A Imidazoline substituted naphthalene compounds for treatment of glaucoma ALLERGAN, INC. (US) 1993-01-19 US claimed
WO-1992021349-A1 COMBINATIONS OF ALPHA-2 ADRENERGIC AGONISTS WITH ALPHA-3 ANTAGONISTS FOR LOWERING INTRAOCULAR PRESSURE ALLERGAN, INC. (US) 1992-12-10 WO claimed
WO-1992011871-A1 STABLE SUSPENSION FORMULATIONS FOR CONTROLLED DELIVERY OF PHARMACEUTICAL COMPOUNDS ALLERGAN, INC. (US) 1992-07-23 WO claimed
WO-1991016869-A1 POLYMERIC DRUG DELIVERY SYSTEM ALLERGAN, INC. (US) 1991-11-14 WO claimed
EP-0399791-A1 Combinations of selective alpha-adrenergic agonists and antagonists useful in lowering intraocular pressure ALLERGAN, INC (US) 1990-11-28 EP claimed
CN-114173793-A Composition, kit and use thereof 泰瑞威公司 2022-03-11 CN disclosed
CN-114080220-A Method for preparing gel-forming composition 泰瑞威公司 2022-02-22 CN disclosed
CN-113825498-A Improved lyophilized formulations comprising hyaluronic acid and plasma proteins and uses thereof 骨治疗公司 2021-12-21 CN disclosed
WO-1991016869-A1 POLYMERIC DRUG DELIVERY SYSTEM ALLERGAN, INC. (US) 1991-11-14 WO disclosed
US-5021410-A Administering hypotensive agent to the eye of a mammal ALLERGAN, INC. (US) 1991-06-04 US disclosed
EP-0399791-A1 Combinations of selective alpha-adrenergic agonists and antagonists useful in lowering intraocular pressure ALLERGAN, INC (US) 1990-11-28 EP disclosed