SCHEMBL5650776

SCHEMBL5650776

COc1cc2c(Nc3cnc(NC(=O)c4cccc(Cl)c4)nc3)ncnc2cc1OCc1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AURKA O14965 6/20 0.71
KDR P35968 5/20 0.70
EGFR P00533 9/20 0.69
AURKB Q96GD4 5/20 0.61
MAPK14 Q16539 3/20 0.60
IRAK4 Q9NWZ3 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10152557 0.93 AURKA (0.69) AURKAKDREGFRAURKBMAPK14
SCHEMBL5651656 0.92 EGFR (0.65) AURKAKDREGFRAURKBMAPK14
Hydrochloric Acid SCHEMBL2063014 0.92 AURKA (0.69) AURKAKDREGFRAURKBMAPK14
Hydrochloric Acid SCHEMBL5652341 0.92 AURKA (0.69) AURKAKDREGFRAURKBMAPK14
SCHEMBL5022265 0.91 KDR (0.70) AURKAKDREGFRAURKBMAPK14
SCHEMBL5016618 0.90 AURKA (0.69) AURKAKDREGFRAURKBMAPK14
SCHEMBL5023489 0.89 AURKA (0.78) AURKAKDREGFRAURKBMAPK14
SCHEMBL5091097 0.88 AURKA (0.70) AURKAKDREGFRAURKBMAPK14
SCHEMBL5655354 0.88 EGFR (0.65) AURKAKDREGFRAURKBMAPK14
SCHEMBL5653702 0.87 AURKA (0.71) AURKAKDREGFRAURKBMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7235559-B1 Therapeutic quinazoline derivatives ASTRAZENECA AB (SE) 2007-06-26 US disclosed