SCHEMBL5651444

SCHEMBL5651444

O=C(NN1CCCCC1)c1ccc(-c2nc3ncccc3[nH]2)cc1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 1/20 0.59
AURKA O14965 5/20 0.59
HPSE Q9Y251 2/20 0.56
HTT P42858 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5653824 0.83 AURKA (0.45) PRMT5AURKAHPSEHTT
SCHEMBL5650901 0.83 AURKA (0.45) PRMT5AURKAHPSEHTT
SCHEMBL5653967 0.83 AURKA (0.45) PRMT5AURKAHPSEHTT
SCHEMBL5651334 0.81 HPSE (0.57) HPSEHTT
SCHEMBL5651844 0.81 PDE2A (0.56) PRMT5AURKA
SCHEMBL5652807 0.80 PDE5A (0.53) AURKAHTT
SCHEMBL5654880 0.80 AURKA (0.45) PRMT5AURKAHPSEHTT
SCHEMBL5651534 0.79 HTT (0.52) HPSEHTT
SCHEMBL14022277 0.77 PRMT5 (0.67) PRMT5AURKAHPSE
SCHEMBL6265479 0.76 HPSE (0.65) PRMT5AURKAHPSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7220769-B2 Azolylbenzamides and analogues and their use for treating osteoporosis NIKEM RESEARCH S.R.L. (IT) 2007-05-22 US disclosed
US-20050038095-A1 Azolylbenzamides and analogues and their use for treating osteoporosis 3-V BIOSCIENCES, INC. 2005-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050038095-A1 Azolylbenzamides and analogues and their use for treating osteoporosis NR0B2, NR0B1, NCOR1 PRMT5 448/4885AURKA 4787/4885HPSE 3728/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.