SCHEMBL5653181

SCHEMBL5653181

CCCn1c(=O)c2c(nc(Cc3ccnnc3)n2CCN(CC)CCO)n(CCc2cc(NC(C)=O)ccc2O)c1=O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.41
ALDH1A1 P00352 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 2/20 0.36
ADORA2B P29275 6/20 0.35
RXFP1 Q9HBX9 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPC1 O15118 1/20 0.32
GAA P10253 1/20 0.32
RAB9A P51151 1/20 0.32
ADORA3 P0DMS8 2/20 0.31
PDE4B Q07343 1/20 0.31
MAPK1 P28482 1/20 0.30
CYP3A4 P08684 1/20 0.30
ADORA2A P29274 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1334411 0.91 ADORA1 (0.42) ADORA1ALDH1A1KMT2ASMN1; SMN2TSHR
SCHEMBL5653185 0.89 ADORA1 (0.43) ADORA1ALDH1A1KMT2ASMN1; SMN2TSHR
SCHEMBL1334722 0.81 ADORA1 (0.49) ADORA1ALDH1A1KMT2ASMN1; SMN2TSHR
SCHEMBL1334414 0.80 ADORA1 (0.44) ADORA1ALDH1A1KMT2ASMN1; SMN2TSHR
SCHEMBL1333023 0.79 ADORA1 (0.50) ADORA1ALDH1A1KMT2ASMN1; SMN2TSHR
SCHEMBL1334330 0.78 ADORA1 (0.44) ADORA1ALDH1A1KMT2ASMN1; SMN2TSHR
SCHEMBL5044751 0.77 ADORA1 (0.48) ADORA1ALDH1A1KMT2ASMN1; SMN2TSHR
SCHEMBL1333466 0.77 ADORA1 (0.47) ADORA1ALDH1A1KMT2ASMN1; SMN2TSHR
SCHEMBL4167581 0.74 ADORA1 (0.44) ADORA1ALDH1A1KMT2ASMN1; SMN2TSHR
SCHEMBL1334308 0.74 ADORA1 (0.57) ADORA1ALDH1A1SMN1; SMN2TSHRADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247639-B2 A1 adenosine receptor antagonists ENDACEA, INC. (US) 2007-07-24 US claimed