SCHEMBL5653766

SCHEMBL5653766

COC1=CC(=O)C(Nc2ncnc3cc(OCC4CCN(C)CC4)c(OC)cc23)=CC1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 12/20 1.00
SRC P12931 2/20 0.64
EGFR P00533 12/20 0.63
FGFR1 P11362 4/20 0.63
FLT1 P17948 4/20 0.63
FLT4 P35916 4/20 0.63
BMPR1B O00238 1/20 0.61
PLK4 O00444 1/20 0.61
CIT O14578 1/20 0.61
GAK O14976 1/20 0.61
EPHB6 O15197 1/20 0.61
RIPK2 O43353 1/20 0.61
ROCK2 O75116 1/20 0.61
STK10 O94804 1/20 0.61
MAP4K4 O95819 1/20 0.61
ABL1 P00519 1/20 0.61
ERBB2 P04626 1/20 0.61
LCK P06239 1/20 0.61
FYN P06241 1/20 0.61
CSF1R P07333 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5651242 0.94 KDR (0.89) KDRSRCEGFRFGFR1FLT1
SCHEMBL5654784 0.91 KDR (1.00) KDRSRCEGFRFGFR1FLT1
SCHEMBL5652553 0.90 KDR (0.82) KDRSRCEGFRFGFR1FLT1
SCHEMBL5648069 0.90 KDR (1.00) KDREGFR
SCHEMBL5648809 0.89 KDR (0.82) KDREGFR
SCHEMBL5648208 0.86 KDR (1.00) KDRSRCEGFR
SCHEMBL5652926 0.83 KDR (0.71) KDRSRCEGFR
SCHEMBL5651670 0.83 KDR (0.82) KDREGFR
SCHEMBL5651095 0.83 KDR (0.73) KDR
SCHEMBL5650601 0.82 KDR (0.71) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070299092-A1 Quinone Substituted Quinazoline and Quinoline Kinase Inhibitors WYETH (US) 2007-12-27 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070299092-A1 Quinone Substituted Quinazoline and Quinoline Kinase Inhibitors KDR, FLT1, FLT4 KDR 1/4885SRC 960/4885EGFR 439/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.