SCHEMBL5655522

SCHEMBL5655522

Fc1cc(C2=NO[C@H](COc3ccon3)C2)ccc1-n1cccn1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MIF P14174 13/20 0.36
LMNA P02545 2/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5655513 1.00 MIF (0.36) MIFLMNAMAPTKDM4EACHE
SCHEMBL5654955 0.87 MIF (0.36) MIFLMNAMAPTKDM4E
SCHEMBL5654962 0.87 MIF (0.36) MIFLMNAMAPTKDM4E
SCHEMBL5657087 0.87 MIF (0.39) MIFLMNAMAPTKDM4E
SCHEMBL5657092 0.87 MIF (0.39) MIFLMNAMAPTKDM4E
SCHEMBL5654816 0.85 MIF (0.36) MIFLMNAMAPTKDM4E
SCHEMBL5654812 0.85 MIF (0.36) MIFLMNAMAPTKDM4E
SCHEMBL5654502 0.84 MIF (0.36) MIFLMNAMAPTKDM4E
SCHEMBL5654496 0.84 MIF (0.36) MIFLMNAMAPTKDM4E
SCHEMBL5655145 0.82 PDE3B (0.42) MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070281916-A1 Substituted isoxazolines and their use as antibacterial agents ASTRAZENECA AB (SE) 2007-12-06 US disclosed
US-7081538-B1 Substituted isoxazolines and their use as antibacterial agents ASTRAZENECA AB (SE) 2006-07-25 US disclosed
EP-1242416-B1 SUBSTITUTED ISOXAZOLINES AND THEIR USE AS ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2005-04-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070281916-A1 Substituted isoxazolines and their use as antibacterial agents CYP2S1, CYP3A7, CYP3A5 MIF 4704/4885LMNA 2157/4885MAPT 4743/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.