SCHEMBL5659844

SCHEMBL5659844

Cc1ccc(C2(c3cc(C)c(O)c(C)c3)C(=O)N(c3cccc(OC(F)(F)F)c3)c3ccccc32)c(O)c1C

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 1/20 0.33
POLB P06746 1/20 0.33
RECQL P46063 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
EDNRB P24530 1/20 0.32
EDNRA P25101 1/20 0.32
CCKBR P32239 1/20 0.32
CETP P11597 10/20 0.32
AMPD2 Q01433 1/20 0.32
TRPC5 Q9UL62 1/20 0.31
TOP2A P11388 1/20 0.31
NPY5R Q15761 1/20 0.31
PDE10A Q9Y233 1/20 0.31
GPR142 Q7Z601 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5661607 0.94 OPRL1 (0.33) OPRL1EDNRBEDNRACCKBRCETP
SCHEMBL5657669 0.89 MAPT (0.39) POLBRECQLNPSR1TDP1
SCHEMBL5660992 0.86 OPRL1 (0.35) OPRL1EDNRBEDNRACCKBRCETP
SCHEMBL5659702 0.86 NPSR1 (0.37) POLBRECQLNPSR1TDP1
SCHEMBL5659652 0.84 CETP (0.34) OPRL1EDNRBEDNRACCKBRCETP
SCHEMBL5656691 0.83 SCN9A (0.37) OPRL1EDNRBEDNRACCKBRCETP
SCHEMBL5658788 0.82 MAPT (0.38) POLB
SCHEMBL5656443 0.79 MAPT (0.44)
SCHEMBL5659537 0.79 SLC6A2 (0.36) POLBNPSR1TDP1
SCHEMBL5663116 0.79 SLC6A2 (0.36) POLBNPSR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7250442-B2 Dihydroindol-2-one derivatives as steroid hormone nuclear receptor modulators ELI LILLY AND COMPANY (US) 2007-07-31 US disclosed
US-7250442-B2 Dihydroindol-2-one derivatives as steroid hormone nuclear receptor modulators ELI LILLY AND COMPANY (US) 2007-07-31 US disclosed
US-7250442-B2 Dihydroindol-2-one derivatives as steroid hormone nuclear receptor modulators ELI LILLY AND COMPANY (US) 2007-07-31 US disclosed
US-20050054712-A1 Dihydroindol-2-one derivatives as steroid hormone nuclear receptor modulators ELI LILLY AND COMPANY 2005-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050054712-A1 Dihydroindol-2-one derivatives as steroid hormone nuclear receptor modulators NR3C2, NR5A1, NR5A2 OPRL1 267/4885POLB 4753/4885RECQL 3363/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.